SCHEMBL6933926

SCHEMBL6933926

CCOC(Cc1ccc(OCCO/N=C(/C)c2ccc(-c3ccccn3)cc2)cc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 18/20 0.55
PPARG P37231 18/20 0.55
PPARD Q03181 11/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6933936 1.00 PPARA (0.55) PPARAPPARGPPARD
SCHEMBL6936505 0.94 PPARG (0.49) PPARAPPARGPPARD
SCHEMBL6936503 0.94 PPARG (0.49) PPARAPPARGPPARD
SCHEMBL6936836 0.92 PPARG (0.47) PPARAPPARGPPARD
SCHEMBL6936834 0.92 PPARG (0.47) PPARAPPARGPPARD
SCHEMBL6933889 0.91 PPARG (0.57) PPARAPPARGPPARD
SCHEMBL6933885 0.91 PPARG (0.57) PPARAPPARGPPARD
SCHEMBL6934112 0.90 PPARG (0.53) PPARAPPARGPPARD
SCHEMBL6934116 0.90 PPARG (0.53) PPARAPPARGPPARD
SCHEMBL6934350 0.90 PPARA (0.64) PPARAPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0916651-B1 PHENYLALKYLCARBOXYLIC ACID DERIVATIVES SANKYO CO (JP) 2003-10-15 EP claimed
US-6103907-A ALDOSE REDUCTASE INHIBITING ANTIDIABETIC AGENT SANKYO COMPANY, LIMITED (JP) 2000-08-15 US claimed
EP-0916651-A1 PHENYLALKYLCARBOXYLIC ACID DERIVATIVES Sankyo Company, Limited (JP) 1999-05-19 EP claimed
EP-0916651-B1 PHENYLALKYLCARBOXYLIC ACID DERIVATIVES SANKYO CO (JP) 2003-10-15 EP disclosed
US-6103907-A ALDOSE REDUCTASE INHIBITING ANTIDIABETIC AGENT SANKYO COMPANY, LIMITED (JP) 2000-08-15 US disclosed
EP-0916651-A1 PHENYLALKYLCARBOXYLIC ACID DERIVATIVES Sankyo Company, Limited (JP) 1999-05-19 EP disclosed