SCHEMBL6933949

SCHEMBL6933949

COCOc1cc(C)cc(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
ACHE P22303 2/20 0.40
CYP1A1 P04798 3/20 0.38
CYP1B1 Q16678 3/20 0.38
MAOB P27338 2/20 0.38
CYP3A4 P08684 2/20 0.37
PTPN1 P18031 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP4B1 P13584 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP3A5 P20815 1/20 0.34
CYP2A7 P20853 1/20 0.34
CYP3A7 P24462 1/20 0.34
CYP2F1 P24903 1/20 0.34
CYP2C18 P33260 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8751846 0.93 KMT2A (0.36) ALDH1A1ACHEMAOBCYP3A4
SCHEMBL2636216 0.91 ALDH1A1 (0.58) ALDH1A1CYP1A1CYP1B1MAOBCYP3A4
SCHEMBL2978585 0.89 ALDH1A1 (0.39) ALDH1A1CYP3A4
SCHEMBL2947790 0.83 ALDH1A1 (0.42) ALDH1A1CYP1A1CYP1B1MAOBCYP1A2
SCHEMBL4604583 0.81 ALDH1A1 (0.46) ALDH1A1ACHECYP1A1CYP1B1MAOB
SCHEMBL12501 0.81 ALDH1A1 (0.73) ALDH1A1ACHECYP1A1CYP1B1CYP3A4
SCHEMBL14461578 0.80 ESR1 (0.52) ALDH1A1ACHECYP1A1CYP1B1MAOB
SCHEMBL4602701 0.79 ALDH1A1 (0.44) ALDH1A1ACHECYP3A4CYP1A2CYP2D6
SCHEMBL12128142 0.79 KCNH2 (0.43) ALDH1A1CYP2A6
SCHEMBL13095988 0.78 ALDH1A1 (0.48) ALDH1A1ACHECYP1A1CYP1B1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9120774-B2 Novobiocin analogues having modified sugar moieties UNIVERSITY OF KANSAS (US) 2015-09-01 US disclosed
US-20120252745-A1 NOVOBIOCIN ANALOGUES HAVING MODIFIED SUGAR MOIETIES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-10-04 US disclosed
US-20110082098-A1 NOVOBIOCIN ANALOGUES AND TREATMENT OF POLYCYSTIC KIDNEY DISEASE UNIVERSITY OF KANSAS (US) 2011-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120252745-A1 NOVOBIOCIN ANALOGUES HAVING MODIFIED SUGAR MOIETIES HSP90AB1, HSP90AB2P, HSP90B1 ALDH1A1 3066/4885ACHE 4861/4885CYP1A1 3699/4885
US-20110082098-A1 NOVOBIOCIN ANALOGUES AND TREATMENT OF POLYCYSTIC KIDNEY DISEASE PKD1, PKD2, HSP90B1 ALDH1A1 4382/4885ACHE 4880/4885CYP1A1 4077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.