SCHEMBL6934133

SCHEMBL6934133

NC(Cc1ccccc1)c1ncc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.47
CYP1A2 P05177 1/20 0.45
EPHX1 P07099 1/20 0.44
MTOR P42345 1/20 0.43
ADK P55263 1/20 0.43
NISCH Q9Y2I1 1/20 0.43
SLC6A2 P23975 2/20 0.41
MAOA P21397 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYP2A6 P11509 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
ROCK2 O75116 1/20 0.40
PRKACA P17612 1/20 0.40
PRKACG P22612 1/20 0.40
PRKACB P22694 1/20 0.40
AKT2 P31751 1/20 0.40
CYP2D6 P10635 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14909320 1.00 TAAR1 (0.47) TAAR1CYP1A2EPHX1MTORADK
SCHEMBL8904389 1.00 TAAR1 (0.47) TAAR1CYP1A2EPHX1MTORADK
SCHEMBL13919511 0.87 LTA4H (0.53) CYP1A2SLC6A2MAOASLC6A3LMNA
SCHEMBL12011595 0.81 NISCH (0.49) TAAR1MTORADKNISCHSLC6A2
SCHEMBL4442877 0.81 TAAR1 (0.49) TAAR1MTORADKNISCHSLC6A2
SCHEMBL7703943 0.80 CYP19A1 (0.40) CYP1A2CYP2A6CYP2D6SMN1; SMN2
SCHEMBL18930740 0.80 CYP19A1 (0.40) CYP1A2CYP2A6CYP2D6SMN1; SMN2
SCHEMBL2872633 0.79 TAAR1 (0.47) TAAR1CYP1A2MTORADKNISCH
SCHEMBL2335773 0.79 TAAR1 (0.47) TAAR1EPHX1MTORADKNISCH
SCHEMBL5693691 0.78 TAAR1 (0.46) TAAR1CYP1A2MTORADKNISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958918-A Novel nicotinamide derivatives or salts thereof FUJIFILM CORP 2013-03-06 CN disclosed
EP-1368449-A1 LIQUID CLEANING COMPOSITIONS AND THEIR USE UNILEVER N.V. (NL) 2003-12-10 EP disclosed
EP-1360268-A1 BLEACHING COMPOSITION OF ENHANCED STABILITY AND A PROCESS FOR MAKING SUCH A COMPOSITION UNILEVER PLC (GB) 2003-11-12 EP disclosed
EP-1319061-A1 LAUNDRY BLEACHING KIT AND METHOD OF BLEACHING A SUBSTRATE UNILEVER PLC (GB) 2003-06-18 EP disclosed
EP-1285055-A1 TARGETED MOIETIES FOR USE IN BLEACH CATALYSTS UNILEVER PLC (GB) 2003-02-26 EP disclosed
EP-1283861-A1 COMPOSITION AND METHOD FOR BLEACHING A SUBSTRATE UNILEVER PLC (GB) 2003-02-19 EP disclosed
EP-1268731-A1 BLEACHING AND DYE TRANSFER INHIBITING COMPOSITION AND METHOD FOR STAIN BLEACHING OF LAUNDRY FABRICS UNILEVER PLC (GB) 2003-01-02 EP disclosed
EP-1259671-A1 METHOD FOR REDUCING DYE FADING OF FABRICS IN LAUNDRY BLEACHING COMPOSITIONS UNILEVER PLC (GB) 2002-11-27 EP disclosed
EP-1240302-A1 BLEACHING COMPOSITION UNILEVER N.V. (NL) 2002-09-18 EP disclosed
EP-1240301-A2 BLEACHING COMPOSITION UNILEVER N.V. (NL) 2002-09-18 EP disclosed
WO-2001064827-A1 COMPOSITION AND METHOD FOR BLEACHING A SUBSTRATE UNILEVER PLC (GB) 2001-09-07 WO disclosed
WO-2001064825-A1 BLEACHING COMPOSITION AND METHOD FOR BLEACHING LAUNDRY FABRICS UNILEVER PLC (GB) 2001-09-07 WO disclosed
WO-2001064994-A1 METHOD FOR REDUCING DYE FADING OF FABRICS IN LAUNDRY BLEACHING COMPOSITIONS UNILEVER PLC (GB) 2001-09-07 WO disclosed
WO-2001064824-A1 BLEACHING AND DYE TRANSFER INHIBITING COMPOSITION AND METHOD FOR STAIN BLEACHING OF LAUNDRY FABRICS UNILEVER PLC (GB) 2001-09-07 WO disclosed
WO-2001048138-A2 BLEACHING COMPOSITION UNILEVER N.V. (NL) 2001-07-05 WO disclosed
WO-2001048137-A1 BLEACHING COMPOSITION UNILEVER N.V. (NL) 2001-07-05 WO disclosed
WO-2001016269-A1 METHOD OF BLEACHING STAINED FABRICS UNILEVER PLC (GB) 2001-03-08 WO disclosed
WO-2001016271-A1 COMPOSITION AND METHOD FOR BLEACHING A SUBSTRATE UNILEVER PLC (GB) 2001-03-08 WO disclosed
WO-2000059461-A1 ORAL COMPOSITION WITH AN IMPROVED TEETH WHITENING EFFECT UNILEVER N.V. (NL) 2000-10-12 WO disclosed
US-5698706-A BLOCKING TUMOR NECROSIS FACTOR CHIROSCIENCE LIMITED (GB) 1997-12-16 US disclosed