SCHEMBL693753

SCHEMBL693753

O=C1CC2CN(Cc3ccccc3)CCN2c2cccc(F)c2N1.O=[N+]([O-])c1c(F)cccc1F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.46
CHRM3 P20309 6/20 0.40
CHRM2 P08172 5/20 0.40
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
BACE1 P56817 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
TACR1 P25103 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015841 0.91 DRD2 (0.53) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2017178 0.91 DRD2 (0.53) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2015062 0.81 DRD2 (0.53) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2013952 0.81 DRD2 (0.53) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL1351177 0.77 DRD2 (0.55) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL691879 0.75 DRD2 (0.48) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2016632 0.75 DRD2 (0.47) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2017655 0.75 DRD2 (0.47) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL2019817 0.72 DRD2 (0.44) DRD2CHRM3CHRM2DRD4DRD3
SCHEMBL691313 0.72 DRD2 (0.47) DRD2CHRM3CHRM2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421870-A2 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2012-02-29 EP disclosed
WO-2010124042-A2 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-10-28 WO disclosed