SCHEMBL6937686

SCHEMBL6937686

COc1ccc2c(c1)C(C)C(C)CC2

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54
CYP19A1 P11511 4/20 0.51
CYP11B1 P15538 1/20 0.51
MTNR1A P48039 4/20 0.49
SIGMAR1 Q99720 2/20 0.49
DRD2 P14416 1/20 0.49
DRD3 P35462 1/20 0.49
CHRNA7 P36544 1/20 0.48
NQO2 P16083 3/20 0.47
MTNR1B P49286 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15095796 0.83 HTR2A (0.51) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL22477091 0.83 HTR2A (0.51) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL805378 0.83 HTR2A (0.51) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL12593301 0.82 HTR2C (0.66) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL13306294 0.82 HTR2C (0.66) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL13306290 0.82 HTR2C (0.66) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL9558526 0.77 HTR2A (0.46) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL9717303 0.77 HTR2A (0.46) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL2463469 0.77 ACHE (0.60) HTR2AHTR2CHTR2BCYP19A1CYP11B1
SCHEMBL269087 0.77 ACHE (0.60) HTR2AHTR2CHTR2BCYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366036-A2 COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF CYTOCHROME P450RAI Allergan, Inc. (US) 2003-12-03 EP disclosed
WO-2002018361-A2 COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF CYTOCHROME P450RAI ALLERGAN, INC. (US) 2002-03-07 WO disclosed