SCHEMBL6940305

SCHEMBL6940305

CC(=O)[C@@H](CCc1cccc(Cl)c1Cl)n1cnc(C(N)=O)c1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADA P00813 13/20 0.72
TAAR1 Q96RJ0 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
JAK3 P52333 1/20 0.34
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939093 0.90 ADA (0.67) ADATAAR1MEN1KMT2A
SCHEMBL6133731 0.84 ADA (1.00) ADA
SCHEMBL6938971 0.83 ADA (0.70) ADATAAR1JAK3
Hydrochloric Acid SCHEMBL6133941 0.83 ADA (0.98) ADA
SCHEMBL6172584 0.77 ADA (0.72) ADA
SCHEMBL6170497 0.75 ADA (0.84) ADA
SCHEMBL6133735 0.73 ADA (0.59) ADATAAR1SCN9A
Hydrochloric Acid SCHEMBL6133945 0.72 ADA (0.58) ADATAAR1SCN9A
SCHEMBL6168422 0.72 ADA (0.68) ADAMEN1KMT2A
SCHEMBL6940309 0.70 ADA (0.53) ADATAAR1JAK3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed