SCHEMBL6940309

SCHEMBL6940309

NC(=O)c1cn(CC(=O)CCCc2cccc(Cl)c2Cl)cn1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADA P00813 8/20 0.53
TAAR1 Q96RJ0 1/20 0.37
FAAH O00519 1/20 0.36
SCN9A Q15858 1/20 0.34
PLA2G4A P47712 1/20 0.34
TNKS O95271 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
RBP4 P02753 1/20 0.33
PNMT P11086 1/20 0.33
KDM5A P29375 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939100 0.87 ADA (0.50) ADATAAR1FAAHSCN9ATNKS
SCHEMBL6133735 0.81 ADA (0.59) ADATAAR1FAAHSCN9ARBP4
Hydrochloric Acid SCHEMBL6133945 0.80 ADA (0.58) ADATAAR1FAAHSCN9ARBP4
SCHEMBL6938975 0.79 ADA (0.52) ADATAAR1FAAHSCN9AKDM5A
SCHEMBL27455357 0.75 TAAR1 (0.53) TAAR1FAAHTNKSTNKS2PARP2
SCHEMBL6172589 0.74 ADA (0.49) ADARBP4KDM5AKDM4CKDM5B
SCHEMBL5067382 0.73 TAAR1 (0.56) ADATAAR1FAAHTNKSTNKS2
SCHEMBL9714098 0.73 LMNA (0.50) ADARBP4KDM5AKDM4CKDM5B
SCHEMBL6170502 0.71 ADA (0.48) ADARBP4KDM5AKDM4CKDM5B
SCHEMBL6940305 0.70 ADA (0.72) ADATAAR1SCN9AJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed