SCHEMBL6941860

SCHEMBL6941860

O=C1Nc2ccccc2/C1=N/Nc1ccc(C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.53
PIM1 P11309 1/20 0.51
AGTR1 P30556 1/20 0.50
LRRK2 Q5S007 3/20 0.49
IDO1 P14902 2/20 0.49
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 2/20 0.47
POLB P06746 2/20 0.47
HSP90AA1 P07900 1/20 0.47
VCP P55072 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
GAA P10253 3/20 0.45
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263628 1.00 KDR (0.53) KDRPIM1AGTR1LRRK2IDO1
SCHEMBL19678415 0.87 LRRK2 (0.58) KDRAGTR1LRRK2IDO1MEN1
SCHEMBL31013507 0.87 LRRK2 (0.58) KDRAGTR1LRRK2IDO1MEN1
SCHEMBL3993251 0.87 LRRK2 (0.58) KDRAGTR1LRRK2IDO1MEN1
SCHEMBL31013508 0.87 LRRK2 (0.58) KDRAGTR1LRRK2IDO1MEN1
SCHEMBL9661928 0.87 LRRK2 (0.58) KDRAGTR1LRRK2IDO1MEN1
SCHEMBL4408992 0.86 MEN1 (0.67) KDRPIM1AGTR1LRRK2IDO1
SCHEMBL4408999 0.86 MEN1 (0.67) KDRPIM1AGTR1LRRK2IDO1
SCHEMBL4895008 0.85 KMT2A (0.52) KDRPIM1AGTR1LRRK2MEN1
SCHEMBL4895014 0.85 KMT2A (0.52) KDRPIM1AGTR1LRRK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030229453-A1 Crystals and structures of PAK4KD kinase PAK4KD SGX PHARMACEUTICALS, INC. 2003-12-11 US disclosed
WO-2003087816-A1 CRYSTALS AND STRUCTURES OF PAK4KD KINASE PAK4KD STRUCTURAL GENOMIX, INC. (US) 2003-10-23 WO disclosed