SCHEMBL4408992

SCHEMBL4408992

O=C1Nc2ccccc2/C1=N/Nc1cccc(C(=O)O)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.67
KMT2A Q03164 5/20 0.67
MAPT P10636 4/20 0.67
L3MBTL1 Q9Y468 3/20 0.67
POLB P06746 2/20 0.67
HSP90AA1 P07900 1/20 0.67
VCP P55072 1/20 0.67
KDR P35968 3/20 0.50
GSK3B P49841 2/20 0.47
LRRK2 Q5S007 2/20 0.46
IDO1 P14902 1/20 0.46
RAB9A P51151 6/20 0.45
NPC1 O15118 5/20 0.45
GAA P10253 3/20 0.45
MCL1 Q07820 2/20 0.45
KDM4E B2RXH2 2/20 0.45
NOX1 Q9Y5S8 1/20 0.45
MAP2K7 O14733 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CDC25B P30305 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4408999 1.00 MEN1 (0.67) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL4409453 0.90 MAPT (0.60) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL4409457 0.90 MAPT (0.60) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL6941860 0.86 KDR (0.53) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL7263628 0.86 KDR (0.53) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL4895014 0.85 KMT2A (0.52) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL4895008 0.85 KMT2A (0.52) MEN1KMT2AMAPTL3MBTL1POLB
SCHEMBL19678415 0.84 LRRK2 (0.58) MEN1KMT2APOLBKDRLRRK2
SCHEMBL3993251 0.84 LRRK2 (0.58) MEN1KMT2APOLBKDRLRRK2
SCHEMBL9661928 0.84 LRRK2 (0.58) MEN1KMT2APOLBKDRLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009135000-A2 INHIBITION OF SHP2/PTPN11 PROTEIN TYROSINE PHOSPHATASE BY NSC-117199 AND ANALOGS H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2009-11-05 WO disclosed