SCHEMBL6941895

SCHEMBL6941895

OC(O)c1cc(N(c2ccccc2)c2ccccc2)ccc1N(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CRHBP P24387 1/20 0.35
ATM Q13315 1/20 0.35
CRHR2 Q13324 1/20 0.35
TLR9 Q9NR96 1/20 0.35
SLC16A3 O15427 1/20 0.31
SLC16A1 P53985 1/20 0.31
APP P05067 1/20 0.30
SLC6A2 P23975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949996 0.80 ALDH1A1 (0.37) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL15511802 0.76 ALDH1A1 (0.50) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL14186205 0.75 ALDH1A1 (0.45) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL10065710 0.75 ALDH1A1 (0.45) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL12304311 0.75 ALDH1A1 (0.45) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL10065558 0.75 ALDH1A1 (0.45) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL19847573 0.74 CA1 (0.36) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL12004561 0.71 ALDH1A1 (0.45) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL12227052 0.70 ALDH1A1 (0.41) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4
SCHEMBL10304824 0.70 ALDH1A1 (0.41) ALDH1A1L3MBTL1KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1164178-B1 Electroluminescent devices having arylamine polymers EASTMAN KODAK CO (US) 2003-09-03 EP disclosed
EP-1164178-A1 Electroluminescent devices having arylamine polymers EASTMAN KODAK COMPANY (US) 2001-12-19 EP disclosed
US-6329086-B1 GOOD SOLUBILITY, EFFICIENCY AND STABILITY; EMITTING COLOR OF THE POLYMER CAN BE EASILY TUNED BY THE INCORPORATION OF DESIRED AROMATIC GROUP; POLYARYLENEVINYLENE EASTMAN KODAK COMPANY 2001-12-11 US disclosed