SCHEMBL6941907

SCHEMBL6941907

COc1ccc(Cc2nc3cnc(N)nc3[nH]2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
CYP2D6 P10635 1/20 0.47
ATM Q13315 1/20 0.47
GRIN1 Q05586 1/20 0.45
GRIN2B Q13224 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.42
CSF1R P07333 2/20 0.42
NTRK2 Q16620 2/20 0.42
NTRK1 P04629 1/20 0.42
NTRK3 Q16288 1/20 0.42
DHFR P00374 2/20 0.42
KMT2A Q03164 1/20 0.42
TYMP P19971 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945088 0.86 CYP1A2 (0.48) CYP2D6POLBLMNAKMT2A
SCHEMBL7077175 0.85 DHFR (0.59) GRIN1GRIN2BDHFR
SCHEMBL4237789 0.83 GRIN1 (0.46) ALDH1A1CYP2D6ATMGRIN1GRIN2B
SCHEMBL6946589 0.81 MAPT (0.37) CYP2D6POLBLMNA
SCHEMBL986239 0.81 GRIN1 (0.47) ALDH1A1CYP2D6ATMGRIN1GRIN2B
SCHEMBL6947942 0.76 EGFR (0.43) CYP2D6POLBDHFR
SCHEMBL13607772 0.75 GRIN1 (0.47) ATMGRIN1GRIN2BNPSR1POLB
SCHEMBL6948621 0.75 PNP (0.47) CYP2D6POLBLMNA
SCHEMBL6950771 0.73 CYP3A4 (0.39) CYP2D6POLBLMNA
SCHEMBL6939915 0.73 DHFR (0.56) LMNADHFRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed