SCHEMBL6942382

SCHEMBL6942382

CC(C)[C@H](NCc1ccc2ccccc2n1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)CN(NC(=O)O)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.42
CTSE P14091 1/20 0.42
PGC P20142 1/20 0.42
CCR1 P32246 1/20 0.42
BACE1 P56817 4/20 0.41
CA2 P00918 2/20 0.41
ADAM17 P78536 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945023 0.90 PSEN1 (0.47) BACE1
SCHEMBL6953685 0.87 CYP3A4 (0.41) CTSDCCR1
SCHEMBL6952143 0.87 CYP3A4 (0.41) CTSDCCR1
SCHEMBL6947796 0.80 CYP3A4 (0.42) CTSDCCR1BACE1ADAM17
SCHEMBL6950300 0.79 CYP3A4 (0.40) CTSDCCR1BACE1
SCHEMBL6946694 0.78 CYP3A4 (0.46) CTSDCCR1BACE1ADAM17
SCHEMBL6953154 0.78 PSEN1 (0.45) BACE1
SCHEMBL6947880 0.78 PSEN1 (0.45) BACE1
SCHEMBL6947903 0.76 CYP3A4 (0.40) CTSDCTSEPGCCCR1
SCHEMBL6712577 0.76 CCR1 (0.50) CCR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633881-B1 AMINE DERIVATIVES OF OXO- AND HYDROXY-SUBSTITUED HYDROCARBONS NARHEX LTD (HK) 2003-10-29 EP claimed
EP-0633881-B1 AMINE DERIVATIVES OF OXO- AND HYDROXY-SUBSTITUED HYDROCARBONS NARHEX LTD (HK) 2003-10-29 EP disclosed