SCHEMBL6942632

SCHEMBL6942632

NC(=O)c1cccc(C(Cc2ccccc2)C(O)C(N)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.49
SLC6A4 P31645 1/20 0.47
FOLH1 Q04609 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
HPGDS O60760 1/20 0.41
PARP1 P09874 6/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MDM2 Q00987 1/20 0.41
PLA2G10 O15496 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2835490 0.75 CYP1A2 (0.53) EPHX1FOLH1TSHRCYP2C19HSD17B10
SCHEMBL262279 0.75 CYP1A2 (0.53) EPHX1FOLH1TSHRCYP2C19HSD17B10
SCHEMBL17064635 0.74 CTSL (0.54) SLC6A4PARP1POLBCYP3A4MAPT
SCHEMBL8521596 0.72 EPHX1 (0.45) EPHX1POLBL3MBTL1ALPIPKM
SCHEMBL8626906 0.72 EPHX1 (0.46) EPHX1SLC6A4PARP1POLBCYP3A4
SCHEMBL6283656 0.72 PARP1 (0.47) SLC6A4PARP1POLBCYP3A4MAPT
SCHEMBL27613443 0.71 PARP1 (0.55) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL28217944 0.71 FOLH1 (0.56) SLC6A4FOLH1PARP1ANPEPENPEP
SCHEMBL8578374 0.70 EPHX1 (0.56) EPHX1POLBL3MBTL1MDM2ANPEP
SCHEMBL28241248 0.70 PARP1 (0.49) SLC6A4OPRM1PARP1POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944582-B1 KETOBENZAMIDES AS CALPAIN INHIBITORS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
EP-0944582-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998025883-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-18 WO disclosed