SCHEMBL6943601

SCHEMBL6943601

COC(=O)C(Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)(N=Cc1ccccc1)C(c1c[nH]cn1)C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 14/20 0.37
NMBR P28336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943557 0.83 SIRT2 (0.41) SIRT2NMBR
SCHEMBL6943596 0.78 SIRT2 (0.44) SIRT2NMBR
SCHEMBL6943605 0.78 SIRT2 (0.44) SIRT2NMBR
SCHEMBL2002152 0.70 SIRT2 (0.48) SIRT2NMBR
SCHEMBL6943555 0.69 SIRT2 (0.49) SIRT2NMBR
SCHEMBL1999641 0.69 SIRT2 (0.49) SIRT2NMBR
SCHEMBL11618667 0.68 SIRT2 (0.54) SIRT2NMBR
SCHEMBL31370665 0.68 SIRT2 (0.48) SIRT2NMBR
SCHEMBL10978566 0.66 SIRT2 (0.48) SIRT2NMBR
SCHEMBL1994628 0.65 SIRT2 (0.49) SIRT2NMBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0928788-B1 Imidazolidin-4-one derivatives useful as anticancer agents PFIZER PROD INC (US) 2003-02-12 EP disclosed
US-6194438-B1 ANTITUMOR AGENTS; ANTICANCER AGENTS; FARNESYL-PROTEIN TRANSFERASE INHIBITOR PFIZER INC. 2001-02-27 US disclosed
US-6174903-B1 INHIBITORS OF THE ENZYME FARNESYL PROTEIN TRANSFERASE AND ARE THEREFORE CAN BE USED AS ANTICANCER AGENT AND ANTITUMOR AGENT PFIZER INC. 2001-01-16 US disclosed
US-6080769-A Imidazolidin-4-one derivatives useful as anticancer agents PFIZER INC. (US) 2000-06-27 US disclosed
EP-1006113-A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use to inhibit abnormal cell growth Pfizer Products Inc. (US) 2000-06-07 EP disclosed
EP-0928788-A1 Imidazolidin-4-one derivatives useful as anticancer agents Pfizer Products Inc. (US) 1999-07-14 EP disclosed