SCHEMBL6944253

SCHEMBL6944253

Cc1c(Oc2ccc(-n3ccnc3)cc2)nc(Cc2ccc3c(c2)OCO3)nc1N(C)CCCN(C)C.Clc1cc(Oc2ccc(-n3ccnc3)cc2)nc(Cc2ccc3c(c2)OCO3)n1

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 18/20 0.73
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
NOS1 P29475 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942111 0.93 NOS2 (0.74) NOS2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6940200 0.92 NOS2 (0.73) NOS2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6942859 0.85 NOS2 (0.73) NOS2
SCHEMBL6946779 0.82 NOS2 (0.61) NOS2
SCHEMBL6940389 0.77 NOS2 (0.61) NOS2
SCHEMBL6939922 0.76 NOS2 (0.59) NOS2
SCHEMBL6940290 0.74 NOS2 (0.57) NOS2
SCHEMBL6941877 0.74 NOS2 (0.54) NOS2NOS1
SCHEMBL6939629 0.74 NOS2 (0.55) NOS2
SCHEMBL6944316 0.74 NOS2 (0.58) NOS2CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268471-B1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS SCHERING AG (DE) 2003-10-15 EP disclosed