Bromide

Bromide

SCHEMBL6944639

Br.O=c1cnnc2ccccc2c1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.48
HTR3A known ✓ P46098 1/20 0.37
ALDH1A1 P00352 3/20 0.48
MAPT P10636 2/20 0.48
HPGD P15428 2/20 0.48
GLA P06280 1/20 0.48
KDM4E B2RXH2 3/20 0.44
CYP1A2 P05177 1/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
MGAM O43451 1/20 0.38
PDE2A O00408 2/20 0.37
PDE3B Q13370 2/20 0.37
PDE3A Q14432 2/20 0.37
NQO2 P16083 1/20 0.37
PDGFRB P09619 2/20 0.34
PDGFRA P16234 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1515043 0.98 ALDH1A1 (0.50) ALDH1A1MAPTHPGDGLAACHE
Hydrochloric Acid SCHEMBL7448684 0.96 ALDH1A1 (0.48) ALDH1A1MAPTHPGDGLAACHE
Hydrochloric Acid SCHEMBL8523156 0.96 ALDH1A1 (0.48) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL17008972 0.86 ALDH1A1 (0.44) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL6999998 0.73 ALDH1A1 (0.50) ALDH1A1MAPTHPGDGLAACHE
Acridine SCHEMBL2401648 0.70 ALDH1A1 (0.94) ALDH1A1MAPTHPGDGLAACHE
Acridine SCHEMBL10801271 0.70 ALDH1A1 (0.94) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL11389056 0.68 KDM4E (0.44) ALDH1A1MAPTHPGDGLAACHE
Acridine SCHEMBL8339 0.67 ALDH1A1 (1.00) ALDH1A1MAPTHPGDGLAACHE
Acridine SCHEMBL29352289 0.67 ALDH1A1 (1.00) ALDH1A1MAPTHPGDGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289966-A1 SUBSTITUTED LACTAMS AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION Bristol-Myers Squibb Pharma Company (US) 2003-03-12 EP disclosed
WO-2001077086-A1 SUBSTITUTED LACTAMS AS INHIBITORS OF Aβ PROTEIN PRODUCTION DUPONT PHARMACEUTICALS COMPANY (US) 2001-10-18 WO disclosed