SCHEMBL6946047

SCHEMBL6946047

O=C(O)C(=O)CC(=O)c1cccc(Cc2cccc(Br)c2)c1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.61
ERCC5 P28715 8/20 0.55
FEN1 P39748 8/20 0.55
HAO1 Q9UJM8 3/20 0.49
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.45
GLA P06280 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7667390 0.93 PTPN1 (0.60) PTPN1ERCC5FEN1HAO1
SCHEMBL6940911 0.88 PTPN1 (0.72) PTPN1ERCC5FEN1HAO1SMN1; SMN2
Dimethylamine SCHEMBL6946035 0.85 PTPN1 (0.68) PTPN1ERCC5FEN1HAO1
SCHEMBL6945130 0.84 FEN1 (0.66) PTPN1ERCC5FEN1HAO1MRGPRX4
SCHEMBL6948181 0.82 PTPN1 (0.61) PTPN1ERCC5FEN1HAO1NPC1
SCHEMBL6951230 0.82 FEN1 (0.77) PTPN1ERCC5FEN1HAO1
SCHEMBL6943572 0.82 PTPN1 (0.69) PTPN1ERCC5FEN1HAO1NPC1
SCHEMBL6951914 0.82 PTPN1 (0.72) PTPN1ERCC5FEN1HAO1NPC1
SCHEMBL6949871 0.81 PTPN1 (0.67) PTPN1ERCC5FEN1HAO1
Dimethylamine SCHEMBL6951644 0.80 FEN1 (0.73) PTPN1ERCC5FEN1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed