SCHEMBL6940911

SCHEMBL6940911

O=C(O)C(=O)CC(=O)c1cccc(Cc2ccccc2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.72
ERCC5 P28715 9/20 0.66
FEN1 P39748 9/20 0.66
HAO1 Q9UJM8 3/20 0.57
PRSS1 P07477 1/20 0.51
PRSS2 P07478 1/20 0.51
PRSS3 P35030 1/20 0.51
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
CES1 P23141 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL6946035 0.97 PTPN1 (0.68) PTPN1ERCC5FEN1HAO1PRSS1
SCHEMBL6949871 0.90 PTPN1 (0.67) PTPN1ERCC5FEN1HAO1PRSS1
SCHEMBL6947604 0.88 ERCC5 (0.61) PTPN1ERCC5FEN1HAO1
SCHEMBL6951230 0.88 FEN1 (0.77) PTPN1ERCC5FEN1HAO1
SCHEMBL6948181 0.88 PTPN1 (0.61) PTPN1ERCC5FEN1HAO1KDM4E
SCHEMBL6946047 0.88 PTPN1 (0.61) PTPN1ERCC5FEN1HAO1SMN1; SMN2
SCHEMBL6943572 0.88 PTPN1 (0.69) PTPN1ERCC5FEN1HAO1KDM4E
SCHEMBL7196671 0.87 ERCC5 (0.66) PTPN1ERCC5FEN1HAO1KDM4E
SCHEMBL7667390 0.86 PTPN1 (0.60) PTPN1ERCC5FEN1HAO1CA1
SCHEMBL6945130 0.86 FEN1 (0.66) PTPN1ERCC5FEN1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed