SCHEMBL6946789

SCHEMBL6946789

c1ccc(CCc2ncc3nc[nH]c3n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.47
IP6K1 Q92551 1/20 0.44
IP6K3 Q96PC2 1/20 0.44
IP6K2 Q9UHH9 1/20 0.44
PIN1 Q13526 1/20 0.43
TAAR1 Q96RJ0 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
QPCT Q16769 7/20 0.40
QPCTL Q9NXS2 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NUDT1 P36639 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29543900 0.86 PDE4A (0.46) HTR2CIP6K1IP6K3IP6K2TAAR1
SCHEMBL434618 0.86 PDE4A (0.46) HTR2CIP6K1IP6K3IP6K2TAAR1
SCHEMBL10602599 0.77 KDM4E (0.37) NPC1RAB9AQPCTKDM4EALDH1A1
SCHEMBL5440110 0.77 CYP1A2 (0.48) IP6K1PIN1ALDH1A1HPGDHSD17B10
SCHEMBL6948806 0.77 JAK2 (0.32) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL1019383 0.75 IP6K1 (0.47) IP6K1RAB9AKDM4EALDH1A1MAPK1
SCHEMBL8332578 0.75 CDK2 (0.50) HTR2CIP6K1IP6K3IP6K2PIN1
SCHEMBL28024950 0.74 HRH3 (0.40) NPC1RAB9AHPGDHRH3
SCHEMBL7158983 0.73 LMNA (0.33) IP6K1KDM4EALDH1A1GLAGAA
SCHEMBL11200729 0.73 KDM4E (0.32) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed
WO-1998039344-A9 NOVEL PURINE INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE 1999-01-21 WO disclosed
WO-1998039344-A1 NOVEL PURINE INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE METABASIS THERAPEUTICS, INC. (US) 1998-09-11 WO disclosed