SCHEMBL694732

SCHEMBL694732

N#CC1(C(N)=O)CC1N1C[C@H](S(=O)(=O)c2ccc(N3CCC(C(F)(F)F)CC3)cc2Cl)C[C@H]1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.41
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL699205 0.89 CTSS (0.44) CTSS
SCHEMBL694301 0.89 CTSS (0.41) CTSS
SCHEMBL695659 0.86 CTSS (0.43) CTSS
SCHEMBL696780 0.86 CTSS (0.40) CTSS
SCHEMBL696447 0.83 CTSS (0.49) CTSS
SCHEMBL695487 0.83 CTSS (0.44) CTSS
Hydrochloric Acid SCHEMBL695250 0.82 CTSS (0.43) CTSS
SCHEMBL695010 0.81 CTSS (0.42) CTSS
SCHEMBL695475 0.81 CTSS (0.43) CTSS
Hydrochloric Acid SCHEMBL695253 0.81 CTSS (0.42) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163793-B2 Proline derivatives HOFFMAN-LA ROCHE INC. (US) 2012-04-24 US claimed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP claimed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO claimed
US-8163793-B2 Proline derivatives HOFFMAN-LA ROCHE INC. (US) 2012-04-24 US disclosed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed