SCHEMBL6947534

SCHEMBL6947534

O=C(O)C(=O)CC(=O)c1cccc(OCc2ccc(F)cc2)c1

nearest known ligand 0.81

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.81
NR4A2 P43354 4/20 0.71
MAOB P27338 3/20 0.66
ERCC5 P28715 1/20 0.59
FEN1 P39748 1/20 0.59
KMT2A Q03164 3/20 0.58
HPD P32754 1/20 0.56
SMPD1 P17405 2/20 0.53
MRGPRX4 Q96LA9 1/20 0.53
MEN1 O00255 2/20 0.53
PPARA Q07869 1/20 0.53
MAOA P21397 1/20 0.53
LMNA P02545 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951340 0.89 PTPN1 (1.00) PTPN1NR4A2MAOBERCC5FEN1
SCHEMBL6946999 0.88 PTPN1 (0.73) PTPN1NR4A2MAOBERCC5FEN1
SCHEMBL1168262 0.84 NR4A2 (1.00) NR4A2MAOBKMT2AHPDMRGPRX4
SCHEMBL6946229 0.81 PTPN1 (0.84) PTPN1NR4A2MAOBERCC5FEN1
SCHEMBL6415086 0.80 MAOB (0.75) NR4A2MAOBKMT2AHPDSMPD1
SCHEMBL4640232 0.80 NR4A2 (0.76) NR4A2MAOBKMT2AHPDMRGPRX4
SCHEMBL6949871 0.79 PTPN1 (0.67) PTPN1ERCC5FEN1LMNA
SCHEMBL6951859 0.79 NR4A2 (0.70) PTPN1NR4A2MAOBKMT2AHPD
SCHEMBL6951854 0.79 NR4A2 (0.70) PTPN1NR4A2MAOBKMT2AHPD
SCHEMBL6131764 0.78 PTPN1 (0.79) PTPN1NR4A2MAOBKMT2ASMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed