SCHEMBL6947698

SCHEMBL6947698

O=C(O)n1cnc2cnc(-c3ccco3)nc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.44
ADORA1 P30542 14/20 0.42
ADORA2A P29274 13/20 0.42
ADORA2B P29275 3/20 0.41
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
PPARG P37231 1/20 0.40
RAB9A P51151 1/20 0.40
NCOA2 Q15596 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
F2 P00734 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942339 0.81 ADORA2A (0.42) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL6948678 0.78 ADORA2A (0.41) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL3267606 0.70 ADORA2A (0.56) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL3270277 0.70 ADORA2A (0.76) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL11780649 0.68 ADORA3 (0.51) ADORA3ADORA1ADORA2AADORA2BMAPT
SCHEMBL3275170 0.68 ADORA2A (0.73) ADORA3ADORA1ADORA2AADORA2BMAPT
SCHEMBL22573814 0.67 ADORA3 (0.56) ADORA3ADORA1ADORA2AADORA2BMAPT
SCHEMBL3273966 0.66 ADORA2A (0.59) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL3273958 0.65 ADORA2A (0.56) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9352344 0.65 POLB (0.46) ADORA3ADORA1ADORA2AADORA2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed