SCHEMBL6947859

SCHEMBL6947859

O=C(O)C(=O)CC(=O)c1cccc(Cc2c(F)c(F)c(F)c(F)c2F)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.67
FEN1 P39748 11/20 0.54
ERCC5 P28715 10/20 0.54
HAO1 Q9UJM8 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946155 0.89 PTPN1 (0.76) PTPN1FEN1ERCC5HAO1
SCHEMBL6951235 0.86 PTPN1 (0.68) PTPN1FEN1ERCC5HAO1
SCHEMBL6943572 0.84 PTPN1 (0.69) PTPN1FEN1ERCC5HAO1
SCHEMBL6940911 0.83 PTPN1 (0.72) PTPN1FEN1ERCC5HAO1
SCHEMBL6949871 0.83 PTPN1 (0.67) PTPN1FEN1ERCC5HAO1
SCHEMBL6948229 0.83 FEN1 (0.61) PTPN1FEN1ERCC5HAO1
SCHEMBL6947914 0.82 PTPN1 (0.83) PTPN1FEN1ERCC5HAO1
SCHEMBL6947084 0.82 PTPN1 (0.70) PTPN1FEN1ERCC5HAO1
SCHEMBL6945660 0.81 PTPN1 (0.73) PTPN1FEN1ERCC5HAO1
Dimethylamine SCHEMBL6946035 0.81 PTPN1 (0.68) PTPN1FEN1ERCC5HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed