SCHEMBL6948385

SCHEMBL6948385

O=C(O)C(=O)CC(=O)c1cc(Cc2ccccc2)cc(OCc2ccccc2)c1

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.70
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
ERCC5 P28715 5/20 0.50
FEN1 P39748 5/20 0.50
NR4A2 P43354 2/20 0.49
SMPD1 P17405 1/20 0.48
MAOB P27338 2/20 0.47
NR4A1 P22736 1/20 0.46
NR4A3 Q92570 1/20 0.46
HAO1 Q9UJM8 2/20 0.45
SRD5A2 P31213 1/20 0.44
GCK P35557 1/20 0.44
PARP10 Q53GL7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4935528 0.90 PTPN1 (0.79) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL6947067 0.85 PTPN1 (0.53) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL6947604 0.84 ERCC5 (0.61) PTPN1ERCC5FEN1HAO1
SCHEMBL6947647 0.84 PTPN1 (0.70) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL6951325 0.83 PTPN1 (0.49) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL6951340 0.82 PTPN1 (1.00) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL11683646 0.80 PTPN1 (0.72) PTPN1ERCC5FEN1NR4A2MAOB
SCHEMBL6951989 0.80 PTPN1 (0.46) PTPN1MEN1KMT2AERCC5FEN1
SCHEMBL6946229 0.80 PTPN1 (0.84) PTPN1ERCC5FEN1NR4A2SMPD1
SCHEMBL13427458 0.79 MEN1 (0.71) PTPN1MEN1KMT2ANR4A2SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed