SCHEMBL6947604

SCHEMBL6947604

O=C(O)C(=O)CC(=O)c1cc(Cc2ccccc2)cc(Cc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 12/20 0.61
FEN1 P39748 12/20 0.61
PTPN1 P18031 5/20 0.61
HAO1 Q9UJM8 3/20 0.55
PLA2G10 O15496 1/20 0.44
PLA2G2A P14555 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949748 0.89 ERCC5 (0.53) ERCC5FEN1PTPN1HAO1LMNA
SCHEMBL6940911 0.88 PTPN1 (0.72) ERCC5FEN1PTPN1HAO1
SCHEMBL7073904 0.87 TBXAS1 (0.52) ERCC5FEN1PTPN1
SCHEMBL6949384 0.86 ERCC5 (0.46) ERCC5FEN1PTPN1HAO1
SCHEMBL6946089 0.86 HAO1 (0.48) ERCC5FEN1PTPN1HAO1
SCHEMBL6946034 0.85 PTPN1 (0.53) ERCC5FEN1PTPN1HAO1
SCHEMBL6947067 0.85 PTPN1 (0.53) ERCC5FEN1PTPN1HAO1
Dimethylamine SCHEMBL6946035 0.85 PTPN1 (0.68) ERCC5FEN1PTPN1HAO1LMNA
SCHEMBL7671810 0.85 CYP19A1 (0.46) ERCC5FEN1PTPN1HAO1
SCHEMBL6948385 0.84 PTPN1 (0.70) ERCC5FEN1PTPN1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed