SCHEMBL6948569

SCHEMBL6948569

CC(C)c1cc(CC(=O)N2CCOC(CC=O)(c3ccc(Cl)c(Cl)c3)C2)cc(C(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.43
SLC6A2 P23975 6/20 0.36
SLC6A4 P31645 6/20 0.36
TACR2 P21452 2/20 0.35
TACR1 P25103 2/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951632 0.88 KMT2A (0.43) KMT2ASLC6A2SLC6A4TACR2TACR1
SCHEMBL6661492 0.88 KMT2A (0.45) KMT2ASLC6A2SLC6A4TACR2TACR1
SCHEMBL6663095 0.88 KMT2A (0.45) KMT2ASLC6A2SLC6A4TACR2TACR1
SCHEMBL6949126 0.88 KMT2A (0.46) KMT2ASLC6A2SLC6A4TACR2TACR1
SCHEMBL6952753 0.84 KMT2A (0.43) KMT2ASLC6A2SLC6A4TACR1OPRK1
SCHEMBL14028100 0.82 SLC6A4 (0.42) KMT2ASLC6A2SLC6A4
SCHEMBL4941176 0.82 KDM4E (0.43) KMT2ASLC6A2SLC6A4TACR2
SCHEMBL4940368 0.80 KMT2A (0.40) KMT2ASLC6A2SLC6A4TACR2TACR1
SCHEMBL6663404 0.80 TACR2 (0.41) KMT2ATACR2TACR1
Hydrochloric Acid SCHEMBL6946688 0.79 TACR2 (0.41) KMT2ATACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506750-B1 N-(phenylacetyl)morpholine derivatives useful as NK1 receptor antagonists, a process for the preparation thereof, and pharmaceutical compositions containing them as active principle. SANOFI-SYNTHELABO (FR) 2003-01-14 US disclosed