SCHEMBL6948639

SCHEMBL6948639

Cc1ccc(S(=O)(=O)O[C@H]2C[C@@H](O[Si](c3ccccc3)(c3ccccc3)C(C)(C)C)C[C@@H](C(=O)O)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP2D6 P10635 2/20 0.38
TSHR P16473 1/20 0.35
ALDH1A1 P00352 3/20 0.35
TAS2R14 Q9NYV8 1/20 0.34
REN P00797 1/20 0.34
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
RECQL P46063 1/20 0.33
ELANE P08246 1/20 0.33
CA1 P00915 3/20 0.32
CA2 P00918 3/20 0.32
CYP1A2 P05177 1/20 0.32
ENPP3 O14638 1/20 0.31
ENPP1 P22413 1/20 0.31
ENPP2 Q13822 1/20 0.31
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951829 1.00 CYP3A4 (0.41) CYP3A4CYP2C19CYP2D6TSHRALDH1A1
SCHEMBL21987331 0.92 CYP3A4 (0.46) CYP3A4CYP2C19CYP2D6ALDH1A1MEN1
SCHEMBL6950985 0.91 POLB (0.32) CYP3A4CYP2C19TAS2R14POLB
SCHEMBL6946744 0.85 CYP2D6 (0.41) CYP3A4CYP2C19CYP2D6TSHRALDH1A1
SCHEMBL6944375 0.85 CYP2D6 (0.41) CYP3A4CYP2C19CYP2D6TSHRALDH1A1
SCHEMBL6951839 0.85 CYP2D6 (0.41) CYP3A4CYP2C19CYP2D6TSHRALDH1A1
SCHEMBL6949043 0.85 CYP2D6 (0.41) CYP3A4CYP2C19CYP2D6TSHRALDH1A1
SCHEMBL5831935 0.84 BACE1 (0.36) CYP3A4ENPP2
SCHEMBL5831941 0.84 BACE1 (0.36) CYP3A4ENPP2
SCHEMBL25106397 0.83 CYP2D6 (0.46) CYP3A4CYP2C19CYP2D6ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235832-B1 VITAMIN D PRESCURSORS, METHOD AND INTERMEDIATES THERAMEX (MC) 2003-11-19 EP disclosed
EP-1106618-A1 Precursors of the A-ring of vitamin D, and method and intermediates for the preparation thereof LABORATOIRE THERAMEX (MC) 2001-06-13 EP disclosed
US-6191292-B1 ENZYMATIC ESTERIFICATION OF A DIOL, E.G., METHYL-3-ACETOXY-5-HYDROXY-CYCLOHEXANECARBOXYLATE BY A LIPASE AND VINYL ALKANOATE OR AN ACID ANHYDRIDE; CYCLIZATION TO A BICYCLIC(3.1.0)HEXANE DERIVATIVE LABORATOIRE THERAMEX (MC) 2001-02-20 US disclosed