SCHEMBL6950985

SCHEMBL6950985

CC(C)(C)[Si](O[C@H]1C[C@H](OS(=O)(=O)c2ccc(Br)cc2)C[C@H](C(=O)O)C1)(c1ccccc1)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
RORC P51449 3/20 0.31
STS P08842 1/20 0.30
TAS2R14 Q9NYV8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948639 0.91 CYP3A4 (0.41) POLBCYP3A4CYP2C19TAS2R14
SCHEMBL6951829 0.91 CYP3A4 (0.41) POLBCYP3A4CYP2C19TAS2R14
SCHEMBL5831941 0.83 BACE1 (0.36) CYP3A4
SCHEMBL5831935 0.83 BACE1 (0.36) CYP3A4
SCHEMBL21987331 0.82 CYP3A4 (0.46) CYP3A4CYP2C19
SCHEMBL21222072 0.82 BACE1 (0.36) CYP3A4
SCHEMBL22614223 0.82 BACE1 (0.36) CYP3A4
SCHEMBL21222073 0.82 BACE1 (0.36) CYP3A4
SCHEMBL6951863 0.77 BACE1 (0.34)
SCHEMBL6941416 0.76 CHRNA7 (0.43) STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235832-B1 VITAMIN D PRESCURSORS, METHOD AND INTERMEDIATES THERAMEX (MC) 2003-11-19 EP disclosed
EP-1106618-A1 Precursors of the A-ring of vitamin D, and method and intermediates for the preparation thereof LABORATOIRE THERAMEX (MC) 2001-06-13 EP disclosed
US-6191292-B1 ENZYMATIC ESTERIFICATION OF A DIOL, E.G., METHYL-3-ACETOXY-5-HYDROXY-CYCLOHEXANECARBOXYLATE BY A LIPASE AND VINYL ALKANOATE OR AN ACID ANHYDRIDE; CYCLIZATION TO A BICYCLIC(3.1.0)HEXANE DERIVATIVE LABORATOIRE THERAMEX (MC) 2001-02-20 US disclosed