SCHEMBL6949219

SCHEMBL6949219

O=C(O)[C@@H]1C[C@@H](O)C[C@H](OS(=O)(=O)c2ccc(Br)cc2)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.33
CYP2D6 P10635 1/20 0.33
NAAA Q02083 2/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
MMP2 P08253 3/20 0.32
CA12 O43570 1/20 0.32
CA14 Q9ULX7 1/20 0.32
MMP1 P03956 2/20 0.32
MMP9 P14780 2/20 0.32
MMP13 P45452 2/20 0.32
CA2 P00918 2/20 0.32
STS P08842 1/20 0.32
CA1 P00915 1/20 0.32
MMP8 P22894 1/20 0.32
TSHR P16473 1/20 0.32
MMP3 P08254 1/20 0.31
MMP7 P09237 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946798 0.86 CYP2D6 (0.47) CYP2D6POLBCA2CA1TSHR
SCHEMBL6952239 0.86 CYP2D6 (0.47) CYP2D6POLBCA2CA1TSHR
SCHEMBL6952074 0.86 CYP2D6 (0.47) CYP2D6POLBCA2CA1TSHR
SCHEMBL6941416 0.80 CHRNA7 (0.43) STS
SCHEMBL10024491 0.80 CYP2D6 (0.35) CYP2D6NAAALMNAMAPTHTT
SCHEMBL22553706 0.79 CYP2D6 (0.52) CYP2D6NAAAPOLBCA2CA1
SCHEMBL989553 0.79 CYP2D6 (0.52) CYP2D6NAAAPOLBCA2CA1
SCHEMBL6950985 0.75 POLB (0.32) RORCPOLBSTS
SCHEMBL11027801 0.73 CYP2D6 (0.56) CYP2D6NAAALMNAMMP2CA12
SCHEMBL20203253 0.73 CYP2D6 (0.56) CYP2D6NAAALMNAMMP2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235832-B1 VITAMIN D PRESCURSORS, METHOD AND INTERMEDIATES THERAMEX (MC) 2003-11-19 EP disclosed
EP-1106618-A1 Precursors of the A-ring of vitamin D, and method and intermediates for the preparation thereof LABORATOIRE THERAMEX (MC) 2001-06-13 EP disclosed
US-6191292-B1 ENZYMATIC ESTERIFICATION OF A DIOL, E.G., METHYL-3-ACETOXY-5-HYDROXY-CYCLOHEXANECARBOXYLATE BY A LIPASE AND VINYL ALKANOATE OR AN ACID ANHYDRIDE; CYCLIZATION TO A BICYCLIC(3.1.0)HEXANE DERIVATIVE LABORATOIRE THERAMEX (MC) 2001-02-20 US disclosed