SCHEMBL6949288

SCHEMBL6949288

C=CCCn1nc(C(=O)O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 2/20 0.43
PTGER4 P35408 3/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
CNR1 P21554 5/20 0.41
CNR2 P34972 4/20 0.41
MAPT P10636 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25434257 0.92 TSHR (0.48) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6953506 0.87 TSHR (0.41) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6946908 0.85 CYP1A2 (0.52) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5438502 0.82 TSHR (0.54) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31429522 0.82 TSHR (0.54) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3017718 0.81 TSHR (0.53) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30571218 0.80 PARP1 (0.57) TSHRKDM4EHSD17B10CNR1CNR2
SCHEMBL15897852 0.79 TSHR (0.52) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2818345 0.78 CNR1 (0.60) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL19779995 0.77 TSHR (0.56) TSHRCYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829474-B1 INDAZOLE DERIVATIVES HAVING MONOCYCLIC AMINO GROUP NISSHIN SEIFUN GROUP INC (JP) 2003-04-09 EP disclosed
US-6096746-A Indazole compound containing a monocyclic amine structure NISSHIN FLOUR MILLING CO., LTD. (JP) 2000-08-01 US disclosed
US-5945434-A TREATMENT OF GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1999-08-31 US disclosed
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
EP-0829474-A1 INDAZOLE DERIVATIVES HAVING MONOCYCLIC AMINO GROUP NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-03-18 EP disclosed
US-5684003-A GASTROINTESTINAL DISORDERS OR ANTIULCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-11-04 US disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed