SCHEMBL6953506

SCHEMBL6953506

C=CCCn1nc(C(=O)Cl)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CNR1 P21554 8/20 0.40
CNR2 P34972 6/20 0.40
HTR3A P46098 5/20 0.40
PARP1 P09874 1/20 0.40
PTGER4 P35408 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GLS O94925 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949288 0.87 TSHR (0.50) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6946941 0.86 CYP1A2 (0.42) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6954722 0.81 CNR1 (0.50) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL25434257 0.80 TSHR (0.48) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6944701 0.79 CNR1 (0.59) TSHRCNR1CNR2HTR3APARP1
SCHEMBL30571218 0.78 PARP1 (0.57) TSHRCNR1CNR2HTR3APARP1
SCHEMBL6950019 0.78 CYP1A2 (0.45) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6948881 0.78 CNR2 (0.61) TSHRCNR1CNR2HTR3APARP1
SCHEMBL6948381 0.78 CNR1 (0.46) TSHRCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3213906 0.77 PTGER4 (0.61) TSHRCYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829474-B1 INDAZOLE DERIVATIVES HAVING MONOCYCLIC AMINO GROUP NISSHIN SEIFUN GROUP INC (JP) 2003-04-09 EP disclosed
US-6096746-A Indazole compound containing a monocyclic amine structure NISSHIN FLOUR MILLING CO., LTD. (JP) 2000-08-01 US disclosed
US-5945434-A TREATMENT OF GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1999-08-31 US disclosed
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
EP-0829474-A1 INDAZOLE DERIVATIVES HAVING MONOCYCLIC AMINO GROUP NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-03-18 EP disclosed
US-5684003-A GASTROINTESTINAL DISORDERS OR ANTIULCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-11-04 US disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed