SCHEMBL6949822

SCHEMBL6949822

CCOC(=O)CC(NC(=O)CNC(=O)CCCNC(=N)N)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.44
ITGA2B P08514 5/20 0.44
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
ITGAV P06756 4/20 0.40
ITGB6 P18564 4/20 0.40
ITGB5 P18084 3/20 0.40
ROCK2 O75116 1/20 0.37
HTT P42858 1/20 0.36
TBXAS1 P24557 1/20 0.36
ALDH1A1 P00352 4/20 0.35
GAA P10253 3/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
HDAC4 P56524 2/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6952526 0.96 ITGB3 (0.43) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19
SCHEMBL6953427 0.89 ITGB3 (0.45) ITGB3ITGA2BCYP3A4ITGAVITGB6
SCHEMBL7414742 0.87 CYP3A4 (0.47) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19
SCHEMBL6950480 0.87 ITGB3 (0.57) ITGB3ITGA2BITGAVITGB6ITGB5
Hydrochloric Acid SCHEMBL7414735 0.86 CYP3A4 (0.46) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL7414738 0.86 CYP3A4 (0.46) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19
SCHEMBL7393079 0.85 FLT4 (0.41) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19
SCHEMBL6950522 0.85 ITGB3 (0.43) ITGB3ITGA2BROCK2HTTTBXAS1
SCHEMBL4924076 0.84 ITGB3 (0.56) ITGB3ITGA2BITGAVITGB6ITGB5
SCHEMBL7381192 0.83 CYP3A4 (0.55) ITGB3ITGA2BCYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804418-B1 PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-03-26 EP claimed
US-5639765-A OSTEOPOROSIS, PAGET*S DISEASE G. D. SEARLE & CO. (US) 1997-06-17 US claimed
US-5602155-A GUANIDINO ALKYL AND PYRIDINE CARBOXYLATE SUBSTITUTED AMIDES G. D. SEARLE & CO. (US) 1997-02-11 US claimed
WO-1996023771-A2 PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1996-08-08 WO claimed
EP-0804418-B1 PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-03-26 EP disclosed
US-5639765-A OSTEOPOROSIS, PAGET*S DISEASE G. D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5602155-A GUANIDINO ALKYL AND PYRIDINE CARBOXYLATE SUBSTITUTED AMIDES G. D. SEARLE & CO. (US) 1997-02-11 US disclosed
WO-1996023771-A2 PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1996-08-08 WO disclosed