SCHEMBL6950128

SCHEMBL6950128

O=C(O)C(=O)CC(=O)c1cccc(Cc2cc(Cl)ccc2Br)c1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 9/20 0.60
ERCC5 P28715 8/20 0.60
PTPN1 P18031 4/20 0.59
PTGER1 P34995 1/20 0.48
HAO1 Q9UJM8 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.40
MEP1A Q16819 1/20 0.40
MEP1B Q16820 1/20 0.40
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946946 0.88 FEN1 (0.63) FEN1ERCC5PTPN1PTGER1HAO1
SCHEMBL6943744 0.86 PTPN1 (0.75) FEN1ERCC5PTPN1PTGER1HAO1
SCHEMBL6951914 0.85 PTPN1 (0.72) FEN1ERCC5PTPN1HAO1MEN1
SCHEMBL6951230 0.83 FEN1 (0.77) FEN1ERCC5PTPN1HAO1
SCHEMBL6947985 0.81 PTPN1 (0.64) FEN1ERCC5PTPN1PTGER1HAO1
Dimethylamine SCHEMBL6951644 0.81 FEN1 (0.73) FEN1ERCC5PTPN1HAO1
SCHEMBL6947803 0.80 PTPN1 (0.59) FEN1ERCC5PTPN1PTGER1HAO1
SCHEMBL6947650 0.80 PTPN1 (0.72) FEN1ERCC5PTPN1PTGER1HAO1
SCHEMBL6945130 0.79 FEN1 (0.66) FEN1ERCC5PTPN1HAO1MRGPRX4
SCHEMBL6946193 0.79 PTPN1 (0.67) FEN1ERCC5PTPN1HAO1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed