SCHEMBL6943744

SCHEMBL6943744

O=C(O)C(=O)CC(=O)c1cccc(Cc2cc(Cl)ccc2F)c1

nearest known ligand 0.75

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.75
FEN1 P39748 9/20 0.62
ERCC5 P28715 8/20 0.62
PTGER1 P34995 1/20 0.49
HAO1 Q9UJM8 1/20 0.46
SNCA P37840 1/20 0.45
MRGPRX4 Q96LA9 2/20 0.44
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946946 0.89 FEN1 (0.63) PTPN1FEN1ERCC5PTGER1HAO1
SCHEMBL6948227 0.89 PTPN1 (0.77) PTPN1FEN1ERCC5HAO1SNCA
SCHEMBL6950128 0.86 FEN1 (0.60) PTPN1FEN1ERCC5PTGER1HAO1
SCHEMBL7072874 0.86 PTPN1 (1.00) PTPN1FEN1ERCC5HAO1SNCA
SCHEMBL6951230 0.84 FEN1 (0.77) PTPN1FEN1ERCC5HAO1
SCHEMBL6949953 0.84 PTPN1 (0.65) PTPN1FEN1ERCC5HAO1
SCHEMBL6947803 0.83 PTPN1 (0.59) PTPN1FEN1ERCC5PTGER1HAO1
SCHEMBL6945641 0.83 PTPN1 (0.71) PTPN1FEN1ERCC5HAO1
SCHEMBL6946220 0.82 PTPN1 (0.71) PTPN1FEN1ERCC5PTGER1HAO1
SCHEMBL6947914 0.82 PTPN1 (0.83) PTPN1FEN1ERCC5HAO1SNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed