SCHEMBL6950329

SCHEMBL6950329

COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)c2cc(C(C)C)oc12

nearest known ligand 0.88

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 19/20 0.88
PDE4A P27815 18/20 0.88
PDE4B Q07343 18/20 0.88
PDE4C Q08493 18/20 0.88
GFER P55789 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950907 0.89 PDE4D (0.70) PDE4DPDE4APDE4BPDE4C
SCHEMBL6954576 0.89 PDE4D (0.70) PDE4DPDE4APDE4BPDE4C
SCHEMBL7919048 0.87 PDE4D (0.78) PDE4DPDE4APDE4BPDE4CGFER
SCHEMBL6950936 0.86 PDE4D (0.67) PDE4DPDE4APDE4BPDE4C
SCHEMBL7916544 0.86 PDE4D (0.67) PDE4DPDE4APDE4BPDE4C
SCHEMBL8333880 0.86 PDE4D (1.00) PDE4DPDE4APDE4BPDE4C
SCHEMBL6836442 0.85 PDE4D (1.00) PDE4DPDE4APDE4BPDE4C
SCHEMBL14043752 0.84 PDE4D (0.74) PDE4DPDE4APDE4BPDE4CGFER
SCHEMBL5723154 0.83 PDE4D (1.00) PDE4DPDE4APDE4BPDE4CGFER
SCHEMBL13741889 0.83 PDE4D (0.83) PDE4DPDE4APDE4BPDE4CGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193808-A1 Synergistic combination Nycomed GmbH (DE) 2010-06-09 EP disclosed
EP-1849468-A2 Pharmaceutical composition of a pde4 or a pde3/4 inhibitor and a histamine receptor antagonist Nycomed GmbH (DE) 2007-10-31 EP disclosed
WO-2004047817-A1 PDE4 AND PDE3/4 INHIBITORS FOR USE IN THE TREATMENT OF CACHEXIA ALTANA PHARMA AG (DE) 2004-06-10 WO disclosed
EP-0923568-B9 NOVEL BENZOFURAN-4-CARBOXAMIDES ALTANA PHARMA AG (DE) 2003-08-13 EP disclosed
EP-0923568-B1 NOVEL BENZOFURAN-4-CARBOXAMIDES ALTANA PHARMA AG (DE) 2002-12-11 EP disclosed
US-6211203-B1 RESPIRATORY SYSTEM DISORDERS, ANTIINFLAMMATORY AGENTS, ENZYME INHIBITORS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2001-04-03 US disclosed
EP-0923568-A1 NOVEL BENZOFURAN-4-CARBOXAMIDES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-06-23 EP disclosed
WO-1998007715-A9 NOVEL BENZOFURAN-4-CARBOXAMIDES BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-29 WO disclosed
WO-1998007715-A1 NOVEL BENZOFURAN-4-CARBOXAMIDES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-02-26 WO disclosed