SCHEMBL6950803

SCHEMBL6950803

COCc1ccc(Cc2ccccc2)cc1C(=O)CC(=O)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 8/20 0.44
FEN1 P39748 8/20 0.44
HAO1 Q9UJM8 1/20 0.44
HNF4A P41235 1/20 0.43
PTPN1 P18031 6/20 0.43
MPO P05164 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LTC4S Q16873 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN6 P29350 1/20 0.39
TACR1 P25103 1/20 0.38
TACR3 P29371 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948223 0.82 NPC1 (0.47) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6950482 0.80 ERCC5 (0.62) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6946203 0.77 LMNA (0.46) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6950947 0.77 ERCC5 (0.62) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6946227 0.76 ERCC5 (0.47) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6949765 0.76 ERCC5 (0.47) ERCC5FEN1HAO1HNF4APTPN1
Dimethylamine SCHEMBL6947623 0.76 LMNA (0.46) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL5148099 0.76 IDO1 (0.44) ERCC5FEN1HAO1HNF4APTPN1
SCHEMBL6947937 0.75 PTPN1 (0.43) ERCC5FEN1HAO1PTPN1KDM4E
Dimethylamine SCHEMBL6950061 0.75 IDO1 (0.44) ERCC5FEN1HAO1HNF4APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed