SCHEMBL6952425

SCHEMBL6952425

O=C(OCc1ccccc1)N1CCC(c2cc(-c3ccnc4ccccc34)c(-c3ccc(F)cc3)[nH]2)CC1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPC3 Q13507 1/20 0.48
TRPC7 Q9HCX4 1/20 0.48
GRIN2B Q13224 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5726133 0.85 MAPK14 (0.60)
SCHEMBL2662864 0.85 MAPK14 (0.60)
SCHEMBL22589253 0.77 MAPK14 (0.48)
SCHEMBL3099127 0.76 SMN1; SMN2 (0.48) TRPC3TRPC7GRIN2B
SCHEMBL22589139 0.76 MAPK14 (0.48)
SCHEMBL6950656 0.72 CYP2D6 (0.45) GRIN2B
SCHEMBL22589274 0.71 TRPC3 (0.51) TRPC3TRPC7GRIN2B
SCHEMBL22589330 0.71 GRIN2B (0.44) GRIN2B
SCHEMBL22589334 0.70 TRPC3 (0.51) TRPC3TRPC7GRIN2B
SCHEMBL22589172 0.70 TRPC3 (0.51) TRPC3TRPC7GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863757-B1 2-SUBSTITUTED ARYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO INC (US) 2003-03-26 EP disclosed
US-5792778-A TREATMENT OF CYTOKINE MEDIATED DISEASES MERCK & CO., INC. (US) 1998-08-11 US disclosed
WO-1997005877-A1 2-SUBSTITUTED ARYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 1997-02-20 WO disclosed