SCHEMBL695403

SCHEMBL695403

FC(F)(F)c1cnc(OCC2CC3CC3CN2)cn1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.43
CHRNA4 P43681 4/20 0.43
HCRTR1 O43613 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862956 1.00 CHRNB2 (0.43) CHRNB2CHRNA4HCRTR1
SCHEMBL610705 1.00 CHRNB2 (0.43) CHRNB2CHRNA4HCRTR1
SCHEMBL10121582 0.81 HPGD (0.38) CHRNB2CHRNA4HCRTR1
SCHEMBL611439 0.78 CHRNB2 (0.33) CHRNB2CHRNA4
SCHEMBL262092 0.75 HCRTR1 (0.36) CHRNB2CHRNA4HCRTR1
SCHEMBL262093 0.75 HCRTR1 (0.36) CHRNB2CHRNA4HCRTR1
SCHEMBL607998 0.74 NPC1 (0.35) CHRNB2CHRNA4
SCHEMBL21503638 0.71 ALOX5AP (0.34) CHRNB2CHRNA4HCRTR1
SCHEMBL608698 0.68 HPGD (0.36)
SCHEMBL619863 0.67 CHRNB2 (0.38) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421850-A1 3 -AZABICYCLO [4.1.0]HEPTANES USED AS OREXIN ANTAGONISTS Glaxo Group Limited (GB) 2012-02-29 EP disclosed
WO-2010122151-A1 3 -AZABICYCLO [4.1.0] HEPTANES USED AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-10-28 WO disclosed