SCHEMBL6954646

SCHEMBL6954646

N[C@H]1CCc2c(F)cccc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 1.00
DRD3 P35462 8/20 1.00
PLAU P00749 1/20 0.55
HTR6 P50406 1/20 0.48
HTR1A P08908 2/20 0.48
HTR7 P34969 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954655 1.00 DRD2 (1.00) DRD2DRD3PLAUHTR6HTR1A
Hydrochloric Acid SCHEMBL6957062 0.98 DRD2 (0.96) DRD2DRD3PLAUHTR6HTR1A
Hydrochloric Acid SCHEMBL6957052 0.98 DRD2 (0.96) DRD2DRD3PLAUHTR6HTR1A
SCHEMBL22061859 0.85 DRD2 (0.74) DRD2DRD3PLAU
SCHEMBL1239050 0.82 DRD2 (0.70) DRD2DRD3PLAUHTR1AHTR7
SCHEMBL31277853 0.82 DRD2 (0.70) DRD2DRD3PLAUHTR1AHTR7
Hydrochloric Acid SCHEMBL26650591 0.81 DRD2 (0.68) DRD2DRD3PLAUHTR1AHTR7
SCHEMBL4024066 0.79 DRD2 (0.66) DRD2DRD3PLAUHTR6
SCHEMBL16233580 0.79 DRD2 (0.66) DRD2DRD3HTR1AHTR7
SCHEMBL11960186 0.78 DRD2 (0.64) DRD2DRD3PLAUHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757677-B1 BENZOCYCLOHEXYLIMIDAZOLETHIONE DERIVATIVES SYNTEX LLC (US) 2003-06-18 EP disclosed
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed