SCHEMBL695540

SCHEMBL695540

N#CCC(NC(=O)[C@@H]1C[C@@H](S(=O)(=O)c2ccccc2Cl)CN1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.44
CTSC P53634 7/20 0.42
CTSL P07711 4/20 0.42
CTSB P07858 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL695385 0.99 CTSS (0.44) CTSSCTSCCTSLCTSB
Hydrochloric Acid SCHEMBL2107368 0.85 CTSS (0.46) CTSSCTSCCTSLCTSB
SCHEMBL2103633 0.85 CTSS (0.46) CTSSCTSCCTSLCTSB
Hydrochloric Acid SCHEMBL697085 0.81 CTSS (0.56) CTSSCTSLCTSB
SCHEMBL15327130 0.77 CTSS (0.43) CTSSCTSLCTSB
SCHEMBL694969 0.77 CTSS (0.43) CTSSCTSLCTSB
SCHEMBL15327131 0.77 CTSS (0.43) CTSSCTSLCTSB
SCHEMBL702312 0.76 CTSS (0.51) CTSSCTSLCTSB
SCHEMBL697725 0.75 CTSS (0.74) CTSSCTSLCTSB
Hydrochloric Acid SCHEMBL696385 0.75 CTSS (0.50) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP claimed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed