SCHEMBL695731

SCHEMBL695731

CS(=O)(=O)[C@H]1CN[C@H](C(=O)NC2(C#N)CC2)C1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 3/20 0.63
CTSS P25774 16/20 0.57
CTSL P07711 13/20 0.40
CTSB P07858 13/20 0.40
CTSK P43235 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL697466 0.92 CTSS (0.58) CTSCCTSSCTSLCTSBCTSK
SCHEMBL2106602 0.83 CTSC (0.55) CTSCCTSSCTSLCTSBCTSK
Hydrochloric Acid SCHEMBL2105547 0.82 CTSC (0.54) CTSCCTSSCTSLCTSBCTSK
SCHEMBL15193990 0.80 CTSS (0.62) CTSCCTSSCTSLCTSBCTSK
SCHEMBL15194658 0.78 CTSS (0.62) CTSCCTSSCTSLCTSB
SCHEMBL29840821 0.77 CTSC (1.00) CTSCCTSSCTSLCTSBCTSK
SCHEMBL695789 0.77 CTSS (0.63) CTSCCTSSCTSLCTSB
SCHEMBL694339 0.77 CTSS (0.71) CTSCCTSSCTSLCTSB
SCHEMBL696268 0.77 CTSS (0.63) CTSCCTSSCTSLCTSB
Hydrochloric Acid SCHEMBL695404 0.76 CTSS (0.62) CTSCCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed