SCHEMBL695798

SCHEMBL695798

N#Cc1ccccc1CNC(=O)[C@@H]1C[C@@H](S(=O)(=O)c2ccccc2Cl)CN1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.46
P2RX7 Q99572 3/20 0.41
CTSL P07711 4/20 0.41
CTSB P07858 3/20 0.41
EPHX2 P34913 1/20 0.38
PKM P14618 1/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL695516 0.99 CTSS (0.45) CTSSP2RX7CTSLCTSBEPHX2
Hydrochloric Acid SCHEMBL697085 0.83 CTSS (0.56) CTSSCTSLCTSB
SCHEMBL702312 0.78 CTSS (0.51) CTSSCTSLCTSB
Hydrochloric Acid SCHEMBL696385 0.77 CTSS (0.50) CTSSCTSLCTSB
SCHEMBL697725 0.77 CTSS (0.74) CTSSCTSLCTSB
Hydrochloric Acid SCHEMBL694102 0.76 CTSS (0.72) CTSSCTSLCTSB
SCHEMBL694969 0.76 CTSS (0.43) CTSSCTSLCTSBALDH1A1
SCHEMBL15327131 0.76 CTSS (0.43) CTSSCTSLCTSBALDH1A1
SCHEMBL15327130 0.76 CTSS (0.43) CTSSCTSLCTSBALDH1A1
SCHEMBL695867 0.75 CTSS (0.68) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP claimed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed