SCHEMBL6958133

SCHEMBL6958133

NCCc1c(Cl)ccc(Cl)c1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 10/20 0.58
PNMT P11086 1/20 0.43
HTR1A P08908 3/20 0.38
ADRA2A P08913 3/20 0.38
SLC6A2 P23975 3/20 0.38
CYP2C19 P33261 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTR3A P46098 1/20 0.38
BACE1 P56817 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
BLM P54132 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
MAPT P10636 2/20 0.35
ALOX15 P16050 2/20 0.35
DRD1 P21728 2/20 0.35
PTGS1 P23219 2/20 0.35
MAPK1 P28482 2/20 0.35
ADRA1A P35348 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13369610 0.81 CXCR1 (0.44) TAAR1PNMTHTR1AADRA2ASLC6A2
SCHEMBL6953644 0.76 TAAR1 (0.62) TAAR1PNMTCYP3A4TSHRSMN1; SMN2
SCHEMBL11791298 0.73 HSD17B10 (0.39) HTR1AADRA2ASLC6A2CYP2C19KDM4E
SCHEMBL1570203 0.73 TAAR1 (1.00) TAAR1PNMTALDH1A1BACE1DPP4
SCHEMBL13590951 0.73 TAAR1 (0.58) TAAR1PNMTALDH1A1CYP1A2
SCHEMBL5159116 0.72 TAAR1 (0.45) TAAR1PNMTKDM4EBLMKMT2A
SCHEMBL20093628 0.71 HSD17B10 (0.38) HTR1AADRA2ASLC6A2CYP2C19KDM4E
SCHEMBL20103788 0.71 TAAR1 (0.59) TAAR1PNMTBACE1
SCHEMBL3922168 0.70 TAAR1 (0.64) TAAR1PNMTDPP4HSP90AA1ACHE
SCHEMBL2935032 0.68 DPP4 (0.52) CYP2C19ALDH1A1KMT2ATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5714503-A Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 1998-02-03 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
EP-0540143-A2 Compounds and methods for inhibition of HIV and related viruses Medivir Aktiebolag (SE) 1993-05-05 EP disclosed