SCHEMBL6953644

SCHEMBL6953644

NCCc1c(Cl)ccc(Cl)c1Cl

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 8/20 0.62
PNMT P11086 2/20 0.46
MAOB P27338 3/20 0.35
SIGMAR1 Q99720 1/20 0.34
KRAS P01116 1/20 0.34
HRH1 P35367 1/20 0.34
CYP2A6 P11509 1/20 0.33
HTR2A P28223 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103788 0.84 TAAR1 (0.59) TAAR1PNMTMAOBKRAS
SCHEMBL1765193 0.79 PNMT (0.48) TAAR1PNMTCYP2A6HTR2ALOXL2
SCHEMBL1570203 0.77 TAAR1 (1.00) TAAR1PNMTMAOBHTR2ASMN1; SMN2
SCHEMBL6958133 0.76 TAAR1 (0.58) TAAR1PNMTSMN1; SMN2CYP3A4TSHR
SCHEMBL13590951 0.76 TAAR1 (0.58) TAAR1PNMTMAOBKRASCYP2A6
SCHEMBL17552720 0.75 TAAR1 (0.34) TAAR1PNMTCYP2A6SMN1; SMN2CYP3A4
SCHEMBL1005529 0.75 TAAR1 (0.34) TAAR1PNMTCYP2A6CYP3A4
SCHEMBL10830911 0.75 TAAR1 (0.34) TAAR1PNMTCYP2A6CYP3A4
SCHEMBL3414586 0.75 CYP3A4 (0.39) TAAR1SMN1; SMN2CYP3A4TSHR
SCHEMBL10061023 0.75 ALDH1A1 (0.35) TAAR1PNMTSIGMAR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5714503-A Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 1998-02-03 US disclosed
US-5658907-A THIOUREA VIRICIDES MEDIVIR A/B (SE) 1997-08-19 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
EP-0540143-A2 Compounds and methods for inhibition of HIV and related viruses Medivir Aktiebolag (SE) 1993-05-05 EP disclosed
WO-1993003022-A1 COMPOUNDS AND METHODS FOR INHIBITION OF HIV AND RELATED VIRUSES MEDIVIR AB (SE) 1993-02-18 WO disclosed