SCHEMBL6958523

SCHEMBL6958523

Cc1ccc(-c2nc(-c3ccccc3)oc2-c2ccc(C)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.66
RAB9A P51151 6/20 0.66
KDM4E B2RXH2 6/20 0.66
HPGD P15428 5/20 0.66
ALDH1A1 P00352 4/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
MAPT P10636 1/20 0.66
MAPK1 P28482 1/20 0.66
CASP1 P29466 1/20 0.66
CYP2C19 P33261 1/20 0.66
CASP7 P55210 1/20 0.66
ATM Q13315 1/20 0.66
HSD17B10 Q99714 1/20 0.66
NFKB1 P19838 2/20 0.58
NFKB2 Q00653 2/20 0.58
RELA Q04206 2/20 0.58
POLB P06746 2/20 0.58
MAPK13 O15264 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10910380 1.00 NPC1 (0.66) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL14407423 1.00 NPC1 (0.66) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL14195802 0.93 NPC1 (0.56) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL762311 0.89 NR4A2 (0.62) NPC1RAB9AKDM4EHPGDALDH1A1
Dimethylamine SCHEMBL8172161 0.86 MAPK13 (0.56) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL15489590 0.84 NPC1 (0.50) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL9113400 0.83 MAPK14 (0.61) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL14660408 0.83 NR1H4 (0.53) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL8172158 0.82 NOX1 (0.52) NPC1RAB9AKDM4EHPGDALDH1A1
SCHEMBL19700319 0.82 NOX1 (0.52) NPC1RAB9AKDM4EHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095937-B1 Process for the preparation of trisubstituted oxazoles OREAL (FR) 2003-03-12 EP disclosed
US-6333414-B1 BY REACTION OF THIOUREA WITH THE CORRESPONDING DIKETONE ESTER; CARRIED OUT UNDER REACTION CONDITIONS, PARTICULARLY WITH RESPECT TO PH, WHICH ARE INDUSTRIALLY MORE FAVORABLE. L'ORéAL S.A. (FR) 2001-12-25 US disclosed
EP-1095937-A1 Process for the preparation of trisubstituted oxazoles L'OREAL (FR) 2001-05-02 EP disclosed