SCHEMBL6958755

SCHEMBL6958755

COc1c(F)c(F)c(N)c2c(=O)c(C(=O)O)cn(C3(F)CC3)c12

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.44
CACNA1F O60840 1/20 0.41
POLB P06746 1/20 0.41
MAPK1 P28482 1/20 0.41
CACNA1D Q01668 1/20 0.41
KCNH2 Q12809 1/20 0.41
CACNA1S Q13698 1/20 0.41
CACNA1C Q13936 1/20 0.41
TOP2A P11388 1/20 0.40
TOP2B Q02880 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954234 0.86 STAT3 (0.47) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL7471382 0.85 TOP2A (0.44) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL1343268 0.82 GSK3B (0.58) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL6957895 0.81 KCNH2 (0.42) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL500863 0.80 GSK3B (0.64) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL5783269 0.78 GSK3B (0.51) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL502617 0.78 GSK3B (0.51) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL12131079 0.78 GSK3B (0.62) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL8619910 0.77 GSK3B (0.39) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL4671194 0.76 CHRM1 (0.37) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304329-A2 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-23 EP disclosed
EP-0900793-B1 CYCLOALKYLAMINOMETHYLPYRROLIDINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2002-07-24 EP disclosed
US-6194434-B1 MICROBIOCIDES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-02-27 US disclosed
EP-0900793-A1 CYCLOALKYLAMINOMETHYLPYRROLIDINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1999-03-10 EP disclosed
EP-0807630-A1 HETEROCYCLIC COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed