SCHEMBL6957895

SCHEMBL6957895

COc1c(N2CC3CC3(N)C2)c(F)c(N)c2c(=O)c(C(=O)O)cn(C3(F)CC3)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.42
POLB P06746 2/20 0.42
CACNA1F O60840 1/20 0.42
MAPK1 P28482 1/20 0.42
CACNA1D Q01668 1/20 0.42
CACNA1S Q13698 1/20 0.42
CACNA1C Q13936 1/20 0.42
CYP3A4 P08684 1/20 0.38
GSK3B P49841 10/20 0.38
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PRKD3 O94806 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
OPRM1 P35372 1/20 0.34
CLK2 P49760 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967038 0.91 CACNA1F (0.48) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL6957899 0.85 CYP3A4 (0.51) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL6948982 0.84 KCNH2 (0.49) KCNH2POLBCYP3A4KDM4EPRKD3
SCHEMBL6958755 0.81 GSK3B (0.44) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL6973262 0.77 CACNA1F (0.53) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL9023582 0.77 KCNH2 (0.59) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL4677281 0.76 KCNH2 (0.49) KCNH2POLBTOP2AKDM4EALDH1A1
SCHEMBL6009016 0.75 GSK3B (0.52) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL5787321 0.73 CYP3A4 (0.51) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL5787325 0.73 CYP3A4 (0.51) KCNH2POLBCACNA1FMAPK1CACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304329-A2 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-23 EP disclosed
EP-0807630-A1 HETEROCYCLIC COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed