SCHEMBL6958877

SCHEMBL6958877

O=C(O)c1c[nH]c(=S)n1C1CCc2ccc(F)cc2C1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
MAPK1 P28482 1/20 0.34
HDAC8 Q9BY41 2/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
KDM4A O75164 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
AKR1C3 P42330 2/20 0.33
HDAC6 Q9UBN7 1/20 0.33
AKR1C2 P52895 1/20 0.33
PRMT5 O14744 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950305 0.85 GRIN2B (0.40) TDP1AKR1C3
SCHEMBL6959676 0.85 AKR1C3 (0.40) TDP1AKR1C3AKR1C2NPC1ALDH1A1
SCHEMBL6959185 0.85 HTR2B (0.39) TDP1HTR2CHTR2BHDAC8DRD2
SCHEMBL6952411 0.85 TDP1 (0.39) TDP1AKR1C3AKR1C2
SCHEMBL6953224 0.85 TDP1 (0.39) TDP1AKR1C3AKR1C2
SCHEMBL6952484 0.79 HTR2C (0.37) HTR2CHTR2BDRD2HTR2A
SCHEMBL8807404 0.79 HTR2B (0.34) HTR2CHTR2BDRD2HTR2A
SCHEMBL8807409 0.79 HTR2B (0.34) HTR2CHTR2BDRD2HTR2A
SCHEMBL6952490 0.79 HTR2C (0.37) HTR2CHTR2BDRD2HTR2A
SCHEMBL8612852 0.79 TDP1 (0.41) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757677-B1 BENZOCYCLOHEXYLIMIDAZOLETHIONE DERIVATIVES SYNTEX LLC (US) 2003-06-18 EP disclosed