SCHEMBL8612852

SCHEMBL8612852

O=C(O)c1c[nH]c(=S)n1C1Cc2cc(F)cc(F)c2C1

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953224 0.90 TDP1 (0.39) TDP1HCAR2
SCHEMBL6952411 0.90 TDP1 (0.39) TDP1HCAR2
Potassium Ion SCHEMBL8613013 0.88 TDP1 (0.32) TDP1
SCHEMBL8613976 0.87 TDP1 (0.43) TDP1
SCHEMBL8611146 0.83 AKR1C3 (0.33) TDP1
SCHEMBL6958877 0.79 TDP1 (0.45) TDP1
Potassium Ion SCHEMBL6959314 0.78 TDP1 (0.30) TDP1
SCHEMBL8611550 0.75 TDP1 (0.40) TDP1HCAR2
SCHEMBL6954011 0.74 HRH4 (0.40)
SCHEMBL6950349 0.74 HRH4 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed