SCHEMBL6958954

SCHEMBL6958954

CCNc1ncc(Br)cc1C(=O)Nc1ccc(Cl)nc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.47
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
PGK1 P00558 1/20 0.36
SORT1 Q99523 1/20 0.36
LMNA P02545 5/20 0.36
SMN1; SMN2 Q16637 5/20 0.36
ALDH1A1 P00352 4/20 0.36
HTT P42858 3/20 0.36
CHRNA7 P36544 1/20 0.36
MDM4 O15151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743141 0.90 KDR (0.46) KDRHDAC3HDAC4HDAC1HDAC7
SCHEMBL5745351 0.87 KDR (0.40) KDRHDAC3HDAC4HDAC1HDAC7
SCHEMBL5743146 0.81 KDR (0.44) KDRPGK1SORT1LMNACHRNA7
SCHEMBL6952426 0.81 KDR (0.45) KDRLMNASMN1; SMN2ALDH1A1HTT
SCHEMBL4030073 0.78 KDR (0.39) KDRHDAC3HDAC4HDAC1HDAC7
SCHEMBL5746291 0.77 LMNA (0.44) KDRPGK1SORT1LMNACHRNA7
SCHEMBL5746213 0.76 SMN1; SMN2 (0.39) KDRHDAC3HDAC4HDAC1HDAC7
SCHEMBL5746260 0.76 MDM4 (0.44) KDRSORT1SMN1; SMN2ALDH1A1HTT
SCHEMBL5743089 0.75 KDR (0.42) KDRSORT1LMNASMN1; SMN2ALDH1A1
SCHEMBL5746185 0.74 MAPT (0.45) KDRSORT1LMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767172-B1 8-Arylalkyl- and 8-arylheteroalkyl-5, 11-dihydro-6H-dipyrido-[3,2-b:2', 3'-e][1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMA (US) 2003-03-26 EP disclosed
US-5705499-A VIRICIDES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1998-01-06 US disclosed
EP-0767172-A1 8-Arylalkyl- and 8-arylheteroalkyl-5, 11-dihydro-6H-dipyrido-[3,2-b:2', 3'-e][1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1997-04-09 EP disclosed